-
An oligodeoxyribonucleotide containing 5-formyl-2′-deoxycytidine (fC) at the CpG site forms a covalent complex with DNA cytosine-5 methyltransferases (DNMTs)
Kousuke Sato, Kyoji Kawamoto, Shintaro Shimamura, Satoshi Ichikawa and Akira Matsuda*
Bioorg. Med. Chem.. Lett. 2016, 26, 5395-5398.
DOI: 10.1016/j.bmcl.2016.10.040

-
多成分反応を用いた天然物合成と構造活性相関研究
千葉拓也、仲谷岳志、片山勝史、松田彰、市川聡
有機合成化学協会誌 2016, 74, 426-440
-
Revisited Mechanistic Implications of the Joullié −Ugi ThreeComponent Reaction
Akira Katsuyama, Akira Matsuda, and Satoshi Ichikawa*
Org. Lett. 2016, 18, 2552-2555.
DOI: 10.1021/acs.orglett.6b00827

-
Chemical screening identifies EUrd as a novel inhibitor against Temozolomide-resistant glioblastoma-initiating cells.
Yoshihiro Tsukamoto, Naoki Ohtsu, Smile Echizenya, Satoko Otsuguro, Ryosuke Ogura, Manabu Natsumeda, Mizuho Isogawa, Hiroshi Aoki, Satoshi Ichikawa, Masahiro Sakaitani, Akira Matsuda, Katsumi Maenaka, Yukihiko Fujii, Toru Kondo.*
Stem Cells 2016, accepted. DOI: 10.1002/stem.2380
-
Design, Synthesis, and Biological Activity of Isosyringolin A
Shun Kitahata, Takuya Chiba, Takashi Yoshida, Masaki Ri, Shinsuke Iida, Akira Matsuda, and Satoshi Ichikawa*
Org. Lett., 2016, 18, 2312-2315.
DOI: 10.1021/acs.orglett.6b01053

-
Structural insights into inhibition of lipid I production in bacterial cell wall synthesis
Ben, C. Chung, Ellene, H. Mashalidis, Tetsuya, Tanino, Mijung, Kim, Akira, Matsuda, Jiyong, Hong, Satoshi, Ichikawa, Seok-Yong, Lee.*
Nature, 2016, 533, 557-561. DOI: 10.1038/nature17636.

-
Design, synthesis and biological evaluation of a structurally simplified syringoin A Analogues
Takuya, Chiba, Shun, Kitahata, Akira, Matsuda, Satoshi, Ichikawa.*
Chem. Pharm. Bull. 2016, 64, 811-816.

-
Function-Oriented Synthesis: How to Design Simplified Analogues of Antibacterial Nucleoside Natural Products?
Satoshi, Ichikawa*
Chem. Rec. 2016, 16, 1106-1115.
DOI: 10.1002/tcr.201500247
