Laboratory of Drug Discovery, Center for Research and Education on Drug Discovery

Publications

Presented Paper 2017

  1. Impact of Structures of Macrocyclic Michael Acceptors on Covalent Proteasome Inhibition

    Shun Kitahata, Fumika Yakushiji and Satoshi Ichikawa

    Chem. Sci. 20178, 6959-6963.

    DOI: 10.1039/C7SC02941A

    kitahata abst

     

  2. Total Synthesis and Antibacterial Investigation of Plusbacin A3

    Akira Katsuyama, Atmika Paudel, Suresh Panthee, Hiroshi Hamamoto, Toru Kawakami,
    Hironobu Hojo, Fumika Yakushiji and Satoshi Ichikawa

    Org. Lett. 201719, 3771-3774.

    DOI: 10.1021/acs.orglett.7b01629

    勝山さん OL plusbacin A3

     

    OLYMPUS DIGITAL CAMERA

  3. Divergent synthesis of kinase inhibitor derivatives, leading to discovery of selective Gck inhibitors

    Takanori Matsumaru, Makoto Inai, Kana Ishigami, Toshiki Iwamatsu, Hiroshi Maita , Satoko Otsuguro, Takao Nomura, Akira Matsuda, Satoshi Ichikawa, Masahiro Sakaitani, Satoshi Shuto, Katsumi Maenaka, Toshiyuki Kan

    Bioorg. Med. Chem. Lett2017, 27, 2144-2147.

    DOI: 10.1016/j.bmcl.2017.03.055

    松丸さん SAR

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