Laboratory of Drug Discovery, Center for Research and Education on Drug Discovery

Publications

Presented Paper 2021

  1. Probiotic Aspergillus oryzae produces the antitumor mediator and exhibits antitumor effects in pancreatic cancer through p38 MAPK signaling pathway

    Konishi, Hiroaki*; Isozaki, Shotaro; Kashima, Shin; Moriichi, Kentaro; Ichikawa, SatoshiYamamoto Kazuki; Yamamura, Chikage; Ando, Katsuyoshi; Ueno, Nobuhiro; Akutsu, Hiroaki; Ogawa, Naoki; Fujiya, Mikihiro.

    Sci. Rep202111, 1107.

    DOI:10.1038/s41598-021-90707-4

  2. Solid-phase Synthesis of Fluorescent Analogues of Park’s Nucleotide, Lipid I and Lipid II

    Akira Katsuyama, Fumika Yakushiji, Satoshi Ichikawa

    Tetrahedron Lett202173, 153101.

    DOI: 10.1016/j.tetlet.2021.153101

     

  3. Structure, solubility, and permeability relationships in a diverse middle molecule library

    Hiroyuki Miyachi, Kayoko Kanamitsu, Mayumi Ishii, Eri Watanabe, Akira Katsuyama, Satoko Otsuguro
    Fumika Yakushiji, Mizuki Watanabe, Kouhei Matsui, Yukina Sato, Satoshi Shuto, Takashi Tadokoro
    Shunsuke Kita, Takanori Matsumaru, Akira Matsuda, Tomoyasu Hirose, Masato Iwatsuki, Yasuteru Shigeta
    Tetsuo Nagano, Hirotatsu Kojima, Satoshi Ichikawa, Toshiaki Sunazuka, Katsumi Maenaka

    Bioorganic Med. Chem. Lett. 2021, 37, 127847.

    DOI: 10.1016/j.bmcl.2021.127847

     

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