Laboratory of Drug Discovery, Center for Research and Education on Drug Discovery

Publications

Presented Paper 2025

  1. pH-Controlled isomerization kinetics of ortho-disubstituted benzamidines: E/Z isomerism and axial chirality

    Ryota Kimura, Satoshi Ichikawa, Akira Katsuyama

    Beilstein J. Org. Chem. 202521, 1568-1576.

    DOI: 10.3762/bjoc.21.120

  2. Structure–Activity Relationship of Pseudouridimycin Focusing on the Improvement of Chemical Stability

    Ryotaro Okawa, Irina Artsimovitch, Akira Katsuyama, Toyotaka Sato, Courtney C. AldrichSatoshi Ichikawa

    J. Med. Chem. 2025, ASAP

    DOI: 10.1021/acs.jmedchem.5c00052

    大川さん_article

  3. Concise Total Synthesis of Sandramycin and Its Analogues via Cyclodimerization Using Mitsunobu Reaction

    Radhakrishnam R. Ruddarraju, Yuya Komatani, Yasuaki Tokodai, Satoshi Ichikawa

    J. Org. Chem. 202590, 10550−10554

    DOI: 10.1021/acs.joc.5c01067

    Raju_article

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