Member/Research

Results

2014

  • Guanidine bridged nucleic acid (GuNA): an effect of a cationic bridged nucleic acid on DNA binding affinity.
    Shrestha AR, Kotobuki Y,Hari Y, Obika S.
    ChemComm, 50, 575-577 (2014).
  • Intranuclear Aggregation of Mutant FUS/TLS as a Molecular Pathomechanism of Amyotrophic Lateral Sclerosis.
    Nomura T, Watanabe S, Kaneko K, Yamanaka K, Nukina N, Furukawa Y.
    J Biol Chem. 289, 1192-202 (2014)
  • Allosteric regulation of epoxide opening cascades by a pair of epoxide hydrolases in monensin biosynthesis.
    Minami A, Ose T, Sato K, Oikawa A, Kuroki K, Maenaka K, Oguri H, Oikawa H.
    ACS Chem Biol. In the press.
  • Identification of DJ-1-associated regions on human genes from SH-SY5Y cells using chromatin immunoprecipitation sequence technique.
    Yamane, T., Sugimoto, N., Maita, H., Watanabe, K., Takahashi-Niki, K., Maita, C., Kato-Ose, I., Ishikawa, S., Gao, J., Kitaura, H., Niki, T., Iguchi-Ariga, S.M.M. and Ariga, H.
    Journal of Molecular Biology in Press (2014)
  • Rational Hopping of a Peptidic Scaffold into Non-Peptidic Scaffolds: Structurally Novel Potent Proteasome Inhibitors Derived from a Natural Product, Belactosin A.
    Kawamura S, Unno Y, Hirokawa T, Asai A, Arisawa M, Shuto S.
    Chem. Commun. in press.
  • Optimizing the Physicochemical Properties of Raf /MEK Inhibitors by Nitrogen Scanning
    Toshihiro Aoki, Ikumi Hyohdoh, Noriyuki Furuichi, Sawako Ozawa, Fumio Watanabe, Masayuki Matsushita, Masahiro Sakaitani, Kenji Morikami, Kenji Takanashi, Naoki Harada, Yasushi Tomii, Koji Shiraki, Kentaro Furumoto, Mitsuyasu Tabo, Kiyoshi Yoshinari, Kazutomo Ori, Yuko Aoki, Nobuo Shimma, and Hitoshi Iikur
    ACS Medicinal Chemistry Letters, in press. (2014)
  • New Binding Face of C-type Lectin-like Domains
    Hideo Fukuhara, Atsushi Furukawa, Katsumi Maenaka
    Structure (Cell Press), 22, 1694-1696, (2014)


総説、共著など

  • 最新がん薬物療法学―がん薬物療法の最新知見―「その他のセリン・スレオニンキナーゼ阻害薬」
    野口昌幸、堺谷政弘、水津太
    日本臨床、in press. (2014)
  • アカデミア創薬を成功させるために
    長野哲雄、堺谷政弘
    実験医学増刊号、アカデミア創薬の戦略と実例, 羊土社 (2014)
  • 合理的創薬と構造解析
    齊藤貴士、堺谷政弘、前仲勝実
    実験医学増刊号、アカデミア創薬の戦略と実例, 羊土社 (2014)