• 2019
  • 2020
  • 2021
  • 2019年

    1. ・ 2019/10/25 M1 永田さんが 第56回ペプチド討論会において「若手口頭発表賞 Chem.Commun.賞」を受賞しました。おめでとうございます!

    2. ・ Uptake and Metabolism of Mizoribine, an Immunosuppressant, in L5178Y-R Mouse Lymphoma Cells in vitro and Peripheral Blood Mononuclear Cells of Rats and Kidney Transplant Recipients in vivo. K. Oda, N. Mori, M. Okumi, M. Furusa, M. Ishiguro, K.Inoue, S. Shuto, K. Unagami, H. Ishida, K. Tanabe, T. Murakam, Drug Metab. Pharmacokin, 2019, 33, 233-239.

    3. ・ T. Minami, K. Fukuda, N. Hoshiya, H. Fukuda, M. Watanabe, S. Shuto, Synthesis of Enantiomerically Pure 1,2,3-Trisubstituted Cyclopropane Nucleosides Using Pd-Catalyzed Substitution via Directing Group-Mediated C(sp3)?H Activation as a Key Step. Org. Lett., 2019, 21, 656-659.

    4. ・ W. Ichinose, S. M. Cherepanov, A. A. Shabalova, S. Yokoyama, T. Yuhi, H. Yamaguchi, A. Watanabe, Y. Yamamoto, H. Okamoto, S. Horike, J. Terakawa T. Daikoku, M. Watanabe, N. Mano, H. Higashida,* S. Shuto, Development of a Highly Potent Analogue and a Long-Acting Analogue of Oxytocin for the Treatment of Social Impairment-Like Behaviors. J. Med. Chem., 2019, 62, 3297-3310.

    5. ・ Y. Shishido, F. Tomoike, K. Kuwata, H. Fujikawa, Y. Sekido, Y. Murakami-Tonami, T. Kameda, N. Abe, Y. Kimura, S. Shuto, H. Abe, Covalent inhibitor for glutathione S-transferase Pi (GSTP(1?1)) in human cells. ChemBioChem, 2019, 20, 900-905.

    6. ・ S. M. Cherepanov, R. Miura, A. A. Shabalova, W. Ichinose, S. Yokoyama, H. Fukuda, M. Watanabe, H. Higashida, S. Shuto, Synthesis of Oxytocin Derivatives Lipidated via a Carbonate or Carbamate Linkage as a Long-Acting Therapeutic Agent for Social Impairment-Like Behaviors. Bioorg. Med. Chem., 2019, 27, 3358-3363.

    7. ・ M. Sato, H. Aoki-Saito, H. Fukuda, H. Ikeda, Y. Koga, M. Yatomi, H. Tsurumaki, T. Maeno, T. Saito, T. Nakakura, T. Mori, M. Yanagawa, M. Abe, Y. Sako, K. Dobashi, T. Ishizuka, M. Yamada, S. Shuto, T. Hisada, Resolvin E3 attenuates allergic airway inflammation via the interleukin-23/interleukin-17A pathway. FASEB J., 2019, 33, 12750-12759.

    8. ・ K. Yamamoto, T. Tamura, R. Nakamura, S. Suzuki, J. Saito, K. Ueno, S. Shuto, Development of a novel class of peroxisome proliferator-activated receptor (PPAR) gamma ligands as an anticancer agent with a unique binding mode based on a non-thiazolidinedione scaffold. Bioorg. Med. Chem., 2019, 27, 115122-115137.

    9. ・ T. Taniguchi, N. Saito, R. Doi, A. Kimoto, N. Hoshiya, K. Fujiki, S. Shuto, H. Fujioka, M. Arisawa, Y. Sato, Nickel Nanoparticle-Catalyzed Carboxylation of Unsaturated Hydrocarbon with CO2 Using Sulfur-Modified Au-Supported Nickel Material. Chem. Lett., 2019, 48, 1406-1409.

    10. ・ D. Fushihara, H. Fukuda, H. Abe, S. Shuto, Synthesis of 1,1,2-Trisubstituted Cyclopropane Nucleosides in Enantiomerically Pure Forms. Nucleosides, Nucleotides, Nucleic Acids, 2019, 38, 921-941.

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